HPS2280-95
152246-40-7
默认>95%HPLC,若需其他规格请洽询
产品编号 | 规格 | 货期 | 销售价 | 折扣价 | 数量 | 操作 |
---|---|---|---|---|---|---|
HPS2280-95 | 默认>95%HPLC,若需其他规格请洽询 |
25天
|
敬请询价 | 敬请询价 |
|
名字 | Myristoyl-Arg-Lys-Arg-Thr-Leu-Arg-Arg-Leu-OH |
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序列(三字母) | Myristoyl-Arg-Lys-Arg-Thr-Leu-Arg-Arg-Leu-OH |
序列(单字母) | Myr-RKRTLRRL |
CAS# | 152246-40-7 |
分子式 | C₆₀H₁₁₇N₂₁O₁₁ |
分子量 | 1308.72 |
纯度 | 默认>95%HPLC,若需其他规格请洽询 |
合成方法 | Synthetic |
储存条件 | -20 ± 5 °C |
描述 | N-Myristylation provided the octapeptide with an inhibitory activity against protein kinase C (PKC)-catalyzed Ca²⁺ and phosphatidylserine-dependent histone phosphorylation (IC₅₀ = 5 µM). It has been shown that Myr-RKRTLRRL is the first synthetic PKC inhibitor with demonstrated pharmacological activity in intact cells. |