HPS2214-95
729589-58-6
默认>95%HPLC，若需其他规格请洽询
| 产品编号 | 规格 | 货期 | 销售价 | 折扣价 | 数量 | 操作 |
|---|---|---|---|---|---|---|
| HPS2214-95 | 默认>95%HPLC，若需其他规格请洽询 |
25天
|
敬请询价 | 敬请询价 |
 
|
| 名字 | (2-Furoyl)-PAR-2 (2-6)-Orn amide (mouse, rat) trifluoroacetate salt |
|---|---|
| 序列(三字母) | (2-Furoyl)-Leu-Ile-Gly-Arg-Leu-Orn-NH₂ trifluoroacetate salt |
| 序列(单字母) | (2-Furoyl)-LIGRL-Orn-NH₂ |
| CAS# | 729589-58-6 |
| 分子式 | C₃₆H₆₃N₁₁O₈ |
| 分子量 | 777.97 |
| 纯度 | 默认>95%HPLC，若需其他规格请洽询 |
| 合成方法 | Synthetic |
| 储存条件 | -20 ± 5 °C |
| 应用 | Cardiovascular System & Diseases|Hematology |
| 描述 | 2-(2-Furoyl)-PAR-2 (2-6)-Orn amide (mouse, rat) is a potent and selective PAR-2 agonist. In cultured human PAR-2-expressing cells (2-Furoyl)-LIGRLO-amide was equally effective as SLIGRL-amide, in rat PAR-2-expressing cells it was 10 to 25 times more potent than SLIGRLamide in increasing intracellular calcium levels. In bioassays of tissue PAR-2 activity, measured as arterial vasodilation and hyperpolarization this agonist was 10 to 300 times more potent than SLIGRL-amide. |
