HPS1919-95
819048-44-7
默认>95%HPLC,若需其他规格请洽询
产品编号 | 规格 | 货期 | 销售价 | 折扣价 | 数量 | 操作 |
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HPS1919-95 | 默认>95%HPLC,若需其他规格请洽询 |
25天
|
敬请询价 | 敬请询价 |
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名字 | Acetyl-(D-Arg¹⁰,Cys¹¹,D-Phe¹⁴,Cys¹⁷)-β-MSH (10-17) amide trifluoroacetate salt |
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序列(三字母) | Ac-D-Arg-Cys-Glu-His-D-Phe-Arg-Trp-Cys-NH₂ trifluoroacetate salt(Disulfide bond) |
序列(单字母) | Ac-rCEHfRWC-NH₂ |
CAS# | 819048-44-7 |
分子式 | C₅₁H₇₀N₁₈O₁₁S₂ |
分子量 | 1175.3599999999999 |
纯度 | 默认>95%HPLC,若需其他规格请洽询 |
合成方法 | Synthetic |
储存条件 | -20 ± 5 °C |
应用 | Obesity Research|Pituitary & Hypothalamic Hormones |
描述 | Highly potent and selective β-MSH-derived melanocortin-4 receptor (MC-4R) agonist with sub-nanomolar potency. The binding affinities for human MC-4R, MC-1R, MC-3R and MC-5R were 0.55 ± 0.06, 16.78 ± 1.53, 56.79 ± 4.66, and < 500 nM, respectively. Daily subcutaneous injection of this product to diet-induced obese rats over a period of 14 days demonstrated an effect on reduction of fat mass. |